1q8w A 2.2 BS01 peptide B 0 E127 F129 R133 E170 G200 T201 E203 E230 Y235 P236 F239 D328 E114 F116 R120 E157 G187 T188 E190 E217 Y222 P223 F226 D315 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000166,0001669,0001707,0004672,0004674,0004679,0004691,0005515,0005524,0005634,0005737,0005739,0005829,0005886,0005952,0006468,0010737,0016020,0016301,0016310,0016740,0018105,0019904,0031594,0034237,0034605,0036126,0048471,0106310,1904262 P00517 14656443 5 ~ 24 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF 1q8w A 2.2 BS02 M77 A 1 V57 A70 M120 Y122 V123 E170 T183 F327 V44 A57 M107 Y109 V110 E157 T170 F314 D166 K168 E170 N171 D184 T201 D153 K155 E157 N158 D171 T188 2.7.11.11 0000166,0001669,0001707,0004672,0004674,0004679,0004691,0005515,0005524,0005634,0005737,0005739,0005829,0005886,0005952,0006468,0010737,0016020,0016301,0016310,0016740,0018105,0019904,0031594,0034237,0034605,0036126,0048471,0106310,1904262 Kd=5.7uM -logKd/Ki=5.24, Kd=5.7uM IC50=1494nM P00517 14656443 960 SVKEFLAKAKEDFLKKWENPAQNTAHLDQFERIKTLGTGSFGRVMLVKHMETGNHYAMKILDKQKVVKLKQIEHTLNEKRILQAVNFPFLVKLEFSFKDNSNLYMVMEYVPGGEMFSHLRRIGRFSEPHARFYAAQIVLTFEYLHSLDLIYRDLKPENLLIDQQGYIQVTDFGFAKRVKGRTWTLCGTPEYLAPEIILSKGYNKAVDWWALGVLIYEMAAGYPPFFADQPIQIYEKIVSGKVRFPSHFSSDLKDLLRNLLQVDLTKRFGNLKNGVNDIKNHKWFATTDWIAIYQRKVEAPFIPKFKGPGDTSNFDDYEEEEIRVSINEKCGKEFSEF