1ybg A 2.6 BS01 TAV A 1 K22 N23 L26 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 L26 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0007049,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 -logKd/Ki=4.80, Ki=16uM P33038 15701635 550 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 1ybg B 2.6 BS01 TAV B 1 K22 N23 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 R91 A92 I94 W95 P121 H125 G164 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0007049,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 P33038 15701635 650 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 1ybg C 2.6 BS01 TAV C 1 N23 L26 R91 A92 I94 W95 P121 H125 V163 G164 N23 L26 R91 A92 I94 W95 P121 H125 V163 G164 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0007049,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 P33038 15701635 750 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE 1ybg D 2.6 BS01 TAV D 1 K22 N23 R91 A92 I94 W95 P121 H125 V163 G164 F328 K22 N23 R91 A92 I94 W95 P121 H125 V163 G164 F328 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 K22 N23 D49 R91 C115 R120 D305 H334 L370 R371 R397 2.5.1.7 0003824,0005737,0007049,0008360,0008760,0009252,0016740,0016765,0019277,0051301,0071555 -logKd/Ki=4.80, Ki=16uM P33038 15701635 850 MDKFRVQGPTRLQGEVTISGAKNAALPILFAALLAEEPVEIQNVPKLKDIDTTMKLLTQLGTKVERDGSVWIDASNVNNFSAPYDLVKTMRASIWALGPLVARFGQGQVSLPGGCAIGARPVDLHIFGLEKLGAEIKLEEGYVKASVNGRLKGAHIVMDKVSVGATVTIMSAATLAEGTTIIENAAREPEIVDTANFLVALGAKISGQGTDRITIEGVERLGGGVYRVLPDRIETGTFLVAAAISGGKIVCRNAQPDTLDAVLAKLREAGADIETGEDWISLDMHGKRPKAVTVRTAPHPAFPTDMQAQFTLLNLVAEGTGVITETIFENRFMHVPELIRMGAHAEIESNTVICHGVEKLSGAQVMATDLRASASLVLAGCIAEGTTVVDRIYHIDRGYERIEDKLRALGANIERVKGE