2az5 A 2.1 BS01 307 A 1 L57 Y59 S60 Y119 L120 G121 G122 Y151 L43 Y45 S46 Y94 L95 G96 G97 Y126 ? 0005164,0006955,0016020 ic50=22uM -logKd/Ki=5.27, Kd=5.36uM Kd=5360nM, IC50=1300nM P01375 16284179 1 DKPVAHVVANPQAEGQLQWLNLLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az5 B 2.1 BS01 307 A 1 Y59 Y119 L120 G121 Y151 Y50 Y102 L103 G104 Y134 ? 0005164,0006955,0016020 -logKd/Ki=5.27, Kd=5.36uM Kd=5360nM, IC50=1300nM P01375 16284179 1 DKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az5 C 2.1 BS01 307 C 1 L57 Y119 L120 G121 G122 Y151 L43 Y91 L92 G93 G94 Y123 ? 0005164,0006955,0016020 ic50=22uM Kd=5360nM, IC50=1300nM P01375 16284179 2 DKPVAHVVANPQAEGQLQWLNLLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVTKVNLLSAIKSPCPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL 2az5 D 2.1 BS01 307 C 1 Y59 Y119 L120 G121 Y50 Y103 L104 G105 ? 0005164,0006955,0016020 -logKd/Ki=5.27, Kd=5.36uM Kd=5360nM, IC50=1300nM P01375 16284179 2 DKPVAHVVANPQAEGQLQWLNRRANALLANGVELRDNQLVVPSEGLYLIYSQVLFKGQGCPSTHVLLTHTISRIAVSYQTKVNLLSAIKSPCQRAKPWYEPIYLGGVFQLEKGDRLSAEINRPDYLDFAESGQVYFGIIAL