2gbg A 3.0 BS01 1AD A 1 E203 E204 F355 Y548 S631 Y632 Y663 Y667 E166 E167 F318 Y511 S594 Y595 Y626 Y630 Y548 S631 Y632 D709 H741 Y511 S594 Y595 D672 H704 3.4.14.5 0001618,0001662,0001666,0002020,0002337,0002709,0002717,0004177,0004252,0005102,0005518,0005576,0005886,0006508,0007155,0008233,0008236,0008239,0008284,0009986,0010716,0016020,0016324,0016787,0030027,0030139,0030163,0031258,0031295,0033632,0035641,0036343,0042110,0042277,0042802,0042803,0042995,0043542,0045121,0045499,0046581,0046718,0050919,0070161,0090024 -logKd/Ki=7.25, Ki=56nM P14740 16768443 768 RRTYTLADYLKNTFRVKSYSLRWVSDSEYLYKQENNILLFNAEHGNSSIFLENSTFEIFGDSISDYSVSPDRLFVLLEYNYVKQWRHSYTASYSIYDLNKRQLITEEKIPNNTQWITWSQEGHKLAYVWKNDIYVKIEPHLPSHRITSTGKENVIFNGINDWVYEEEIFGAYSALWWSPNGTFLAYAQFNDTGVPLIEYSFYSDESLQYPKTVWIPYPKAGAVNPTVKFFIVNTDSLSSTTTTIPMQITAPASVTTGDHYLCDVAWVSEDRISLQWLRRIQNYSVMAICDYDKTTLVWNCPTTQEHIETSATGWCGRFRPAEPHFTSDGSSFYKIVSDKDGYKHICQFQKDRKPEQVCTFITKGAWEVISIEALTSDYLYYISNEYKEMPGGRNLYKIQLTDHTNKKCLSCDLNPERCQYYSVSLSKEAKYYQLGCRGPGLPLYTLHRSTDQKELRVLEDNSALDKMLQDVQMPSKKLDFIVLNETRFWYQMILPPHFDKSKKYPLLIDVYAGPCSQKADAAFRLNWATYLASTENIIVASFDGRGSGYQGDKIMHAINKRLGTLEVEDQIEAARQFLKMGFVDSKRVAIWGWSYGGYVTSMVLGSGSGVFKCGIAVAPVSRWEYYDSVYTERYMGLPTPEDNLDHYRNSTVMSRAENFKQVEYLLIHGTADDNVHFQQSAQISKALVDAGVDFQAMWYTDEDHGIASSTAHQHIYSHMSHFLQQCFSLR