2igq A 2.0 BS01 ZN A 1 C1031 C1044 C1074 C1078 C56 C69 C99 C103 Y1124 Y1211 Y149 Y230 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 501 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGSCRCGSPKCRHS 2igq A 2.0 BS02 ZN A 2 C1037 C1074 C1080 C1084 C62 C99 C105 C109 Y1124 Y1211 Y149 Y230 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 502 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGSCRCGSPKCRHS 2igq A 2.0 BS03 ZN A 3 C1031 C1033 C1037 C1042 C56 C58 C62 C67 Y1124 Y1211 Y149 Y230 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 503 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGSCRCGSPKCRHS 2igq A 2.0 BS04 ZN A 4 C1172 C1225 C1227 C1232 C191 C241 C243 C248 Y1124 Y1211 Y149 Y230 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 504 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGSCRCGSPKCRHS 2igq A 2.0 BS05 SAH A 1 M1105 W1107 Y1142 R1166 F1167 N1169 H1170 Y1211 C1225 R1226 M130 W132 Y167 R185 F186 N188 H189 Y230 C241 R242 Y1124 Y1211 Y149 Y230 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 IC50=230nM Q9H9B1 20084102 101 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKGSCRCGSPKCRHS 2igq B 2.0 BS01 ZN B 1 C1031 C1044 C1074 C1078 C56 C69 C99 C103 Y1124 Y1211 Y149 Y232 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 501 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKLFSCRCGSPKCRHS 2igq B 2.0 BS02 ZN B 2 C1037 C1074 C1080 C1084 C62 C99 C105 C109 Y1124 Y1211 Y149 Y232 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 502 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKLFSCRCGSPKCRHS 2igq B 2.0 BS03 ZN B 3 C1031 C1033 C1037 C1042 C56 C58 C62 C67 Y1124 Y1211 Y149 Y232 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 503 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKLFSCRCGSPKCRHS 2igq B 2.0 BS04 ZN B 4 C1172 C1225 C1227 C1232 C193 C244 C246 C251 Y1124 Y1211 Y149 Y232 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 Q9H9B1 20084102 504 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKLFSCRCGSPKCRHS 2igq B 2.0 BS05 SAH B 1 M1105 G1106 W1107 S1141 Y1142 R1166 F1167 N1169 H1170 Y1211 C1225 R1226 M130 G131 W132 S166 Y167 R187 F188 N190 H191 Y232 C244 R245 Y1124 Y1211 Y149 Y232 2.1.1.-,2.1.1.367 0002039,0005634,0008270,0016279,0042054,0046974 IC50=230nM Q9H9B1 20084102 102 ERIVSRDIARGYERIPIPCVNAVDSEPCPSNYKYVSQNCVTSPMNIDRNITHLQYCVCIDDCSSSNCMCGQLSMRCWYDKDGRLLPEFNMAEPPLIFECNHACSCWRNCRNRVVQNGLRARLQLYRTRDMGWGVRSLQDIPPGTFVCEYVGELISDSEADVREEDSYLFDLDEVYCIDARFYGNVSRFINHHCEPNLVPVRVFMAHQDLRFPRIAFFSTRLIEAGEQLGFDYGERFWDIKLFSCRCGSPKCRHS