3b8i A 1.9 BS01 OXL A 1 S50 D88 H235 S48 D86 H233 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 G126 R159 V188 M208 I44 G46 G47 S48 D59 D86 D88 T113 E115 A121 F123 G124 R157 V186 M206 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 RASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFGRKSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGAVASDLTASELSKKYTFPEEYQAWARDYMEVK 3b8i B 1.9 BS01 OXL B 1 S50 D88 H235 S48 D86 H233 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 G126 R159 V188 M208 I44 G46 G47 S48 D59 D86 D88 T113 E115 A121 F123 G124 R157 V186 M206 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 RASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFGRKSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGAVASDLTASELSKKYTFPEEYQAWARDYMEV 3b8i C 1.9 BS01 OXL C 1 S50 D88 R159 H235 S48 D86 R157 H233 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 G126 R159 V188 M208 I44 G46 G47 S48 D59 D86 D88 T113 E115 A121 F123 G124 R157 V186 M206 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 RASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFGRKSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGALTASELSKKYTFPEEYQAWARDYME 3b8i D 1.9 BS01 OXL D 1 G48 S50 D88 R159 H235 G46 S48 D86 R155 H231 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 R159 V188 M208 I44 G46 G47 S48 D59 D86 D88 T113 E115 A121 F123 R155 V184 M204 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 RASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFRSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGAVASDLTASELSKKYTFPEEYQAWARDYME 3b8i E 1.9 BS01 OXL E 1 S50 D88 H235 S47 D85 H232 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 G126 R159 V188 M208 I43 G45 G46 S47 D58 D85 D87 T112 E114 A120 F122 G123 R156 V185 M205 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 ASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFGRKSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGAVASDLTASELSKKYTFPEEYQAWARDYMEVK 3b8i F 1.9 BS01 OXL F 1 S50 D88 H235 S48 D86 H233 I46 G48 G49 S50 D61 D88 D90 T115 E117 A123 F125 G126 R159 V188 M208 I44 G46 G47 S48 D59 D86 D88 T113 E115 A121 F123 G124 R157 V186 M206 4.1.1.112 0000287,0003824,0006107,0008948,0016829,0016831,0016833,0019629,0042866,0046421,0046872 Ki=4uM Ki=43000nM Q9HUU1 18081320 288 RASHHELRAMFRALLDSSRCYHTASVFDPMSARIAADLGFECGILGGSVASLQVLAAPDFALITLSEFVEQATRIGRVARLPVIADADHGYGNALNVMRTVVELERAGIAALTIEDTLLPAQFGRKSTDLICVEEGVGKIRAALEARVDPALTIIARTNAELIDVDAVIQRTLAYQEAGADGICLVGVRDFAHLEAIAEHLHIPLMLVTYGNPQLRDDARLARLGVRVVVNGHAAYFAAIKATYDCLREERGAVASDLTASELSKKYTFPEEYQAWARDYMEVK