3dek A 2.4 BS01 RXD A 1 E123 C163 G165 T166 L168 E90 C130 G132 T133 L135 T62 S63 H121 G122 C163 R164 T29 S30 H88 G89 C130 R131 3.4.22.56 0001554,0001666,0001782,0001818,0002020,0004175,0004190,0004197,0004861,0005123,0005515,0005634,0005654,0005737,0005829,0006508,0006915,0006974,0007413,0007507,0007605,0007611,0008047,0008233,0008234,0008627,0009410,0009411,0009611,0009749,0010033,0010038,0010165,0014070,0016005,0016241,0016485,0016787,0021766,0030163,0030182,0030216,0030218,0030220,0030889,0031264,0031647,0032025,0032355,0032496,0034349,0034612,0035094,0035556,0042542,0043025,0043029,0043065,0043200,0043525,0044346,0044877,0045165,0045786,0046007,0048011,0051146,0051384,0051402,0051604,0051716,0061713,0070269,0071310,0071407,0071887,0072734,0097153,0097190,0097193,0097194,0097199,0097200,0140639,1902004,1904019 ic50=27nM -logKd/Ki=7.57, IC50=27nM P42574 18768468 300 DNSYKMDYPEMGLCIIINNKNFHKSTGMTSRSGTDVDAANLRETFRNLKYEVRNKNDLTREEIVELMRDVSKEDHSKRSSFVCVLLSHGEEGIIFGTNGPVDLKKITNFFRGDRCRSLTGKPKLFIIQACRGTELDCGIETKIPVDADFLYAYSTAPGYYSWRNSKDGSWFIQSLCAMLKQYADKLEFMHILTRVNRKVATEFESFSFDATFHAKKQIPCIVSMLTKELYFYH