3f82 A 2.5 BS01 353 A 1 V1092 A1108 K1110 F1124 E1127 M1131 F1134 L1157 M1160 F1200 H1202 M1211 A1221 D1222 F1223 V38 A49 K51 F61 E64 M68 F71 L94 M97 F137 H139 M148 A158 D159 F160 D1204 A1206 R1208 N1209 D1222 D141 A143 R145 N146 D159 2.7.10.1 0004672,0004713,0005524,0006468 Ki=4.6nM -logKd/Ki=8.34, Ki=4.6nM IC50=3.9nM P08581 19260711 2001 LSALNPELVQAVQHVVIGPSSLIVHFNEVIGRGHFGCVYHGTLLKIHCAVKSLNRGEVSQFLTEGIIMKDFSHPNVLSLLGICLRSEGSPLVVLPYMKHGDLRNFIRNETHNPTVKDLIGFGLQVAKGMKFLASKKFVHRDLAARNCMLDEKFTVKVADFGKLPVKWMALESLQTQKFTTKSDVWSFGVLLWELMTRGAPPYPDVNTFDITVYLLQGRRLLQPEYCPDPLYEVMLKCWHPKAEMRPSFSELVSRISAIFSTFIGEHYVHVNATYVNVK