3krj A 2.1 BS01 KRJ A 1 A614 Y665 C666 G669 D670 L785 F797 R801 A71 Y122 C123 G126 D127 L176 F188 R192 D778 A780 R782 N783 D796 N805 D169 A171 R173 N174 D187 N196 2.7.10.1 0004672,0004713,0004714,0005524,0006468,0007169 ic50=1.1nM -logKd/Ki=8.96, IC50=1.1nM P07333,P11362 22039836 923 PKYQVRWKIIESYEGNSYTFIDPTQLPYNEKWEFPRNNLQFGKTLGAGAFGKVVEATAFGLGKEDAVLKVAVKMLKSTAHADEKEALMSELKIMSHLGQHENIVNLLGACTHGGPVLVITEYCCYGDLLNFLRRKRPPGQLSSRDLLHFSSQVAQGMAFLASKNCIHRDVAARNVLLTNGHVAKIGDFGLARDIMNDSNYIVKGARLPVKWMAPESIFDCVYTVQSDVWSYGILLWEIFSLGLNPYPGILVNSKFYKLVKDGYQMAQPAFAPKNIYSIMQACWALEPTHRPTFQQICSFLQEQA