4isk A 1.752 BS01 UMP A 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk A 1.752 BS02 1JY A 1 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk B 1.752 BS01 UMC B 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk B 1.752 BS02 1JY B 1 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk C 1.752 BS01 UMP C 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk C 1.752 BS02 1JY C 1 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk D 1.752 BS01 UMC D 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk D 1.752 BS02 1JY D 1 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk E 1.752 BS01 UMC E 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk E 1.752 BS02 1JY E 1 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk F 1.752 BS01 UMP C 1 R126 R127 R126 R127 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk F 1.752 BS02 UMC F 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk F 1.752 BS03 1JY F 1 H51 I79 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 I79 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 302 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk G 1.752 BS01 UMP G 1 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 C168 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk G 1.752 BS02 1JY G 1 H51 E58 T78 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 H51 E58 T78 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk H 1.752 BS01 UMC H 1 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 R21 C146 Q165 R166 S167 D169 N177 H207 Y209 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 P0A884 23710599 301 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI 4isk H 1.752 BS02 1JY H 1 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 I79 W80 W83 D169 L172 G173 F176 N177 Y209 V262 A263 E58 W80 Y94 C146 R166 D169 P175 E58 W80 Y94 C146 R166 D169 P175 2.1.1.45 0000287,0003723,0004799,0005737,0005829,0006231,0006235,0006417,0008168,0009165,0009314,0016741,0032259,0042803 Ki=1.2nM P0A884 23710599 303 MKQYLELMQKVLDEGTQKNDRTGTGTLSIFGHQMRFNLQDGFPLVTTKRCHLRSIIHELLWFLQGDTNIAYLHENNVTIWDEWADENGDLGPVYGKQWRAWPTPDGRHIDQITTVLNQLKNDPDSRRIIVSAWNVGELDKMALAPCHAFFQFYVADGKLSCQLYQRSCDVFLGLPFNIASYALLVHMMAQQCDLEVGDFVWTGGDTHLYSNHMDQTHLQLSREPRPLPKLIIKRKPESIFDYRFEDFEIEGYDPHPGIKAPVAI