4k5y A 2.977 BS01 1Q5 A 1 F203 M206 L280 N283 T316 L323 Y327 F89 M92 L323 N326 T359 L366 Y370 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 -logKd/Ki=8.17, Kd=6.7nM P00720,P34998 23863939 401 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRPGVYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAFVNEVSRVVFIYFNAFLESFQGFFVSVFACFLNS 4k5y B 2.977 BS01 1Q5 B 1 F203 M206 L280 N283 T316 L320 Y327 F89 M92 L320 N323 T356 L360 Y367 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 P00720,P34998 23863939 401 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAVFIYFNAFLESFQGFFVSVFACFLNS 4k5y B 2.977 BS02 PGW B 1 L135 F138 N157 I232 W236 L21 F24 N43 I275 W279 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 P00720,P34998 23863939 502 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAVFIYFNAFLESFQGFFVSVFACFLNS 4k5y B 2.977 BS03 PGW B 2 C128 I129 V132 A133 V136 L140 C14 I15 V18 A19 V22 L26 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 P00720,P34998 23863939 503 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAVFIYFNAFLESFQGFFVSVFACFLNS 4k5y B 2.977 BS04 PGW B 3 H199 Y270 Q273 M276 A277 L280 F284 Y327 H85 Y310 Q313 M316 A317 L320 F324 Y367 E1011 D1020 E116 D125 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 P00720,P34998 23863939 504 HYHVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTNIFEMLRIDEGLRLKIYKDTEGYYTIGIGHLLTKSPSLSVAKSELDKAIGRNSNGVITKDEAEKLFNQDVDAAVRGILRNAKLKPVYDSLDAVRRSALINMVFQMGETGVAGFTNSLRMLQQKRWDEAAVNLAKSRWYNQTPNRAKRVIATFRTGTWDAYDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAVFIYFNAFLESFQGFFVSVFACFLNS 4k5y C 2.977 BS01 1Q5 C 1 F203 M206 G210 L280 N283 F284 T316 L320 L323 Y327 F87 M90 G94 L161 N164 F165 T197 L201 L204 Y208 ?,3.2.1.17 0003796,0003824,0004888,0004930,0007166,0007186,0008152,0009253,0016020,0016787,0016798,0016998,0030430,0031640,0042742,0044659 P00720,P34998 23863939 401 HVAAIINYLGHCISLVALLVAFVLFLRARSIRCLRNIIHANLIAAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTDRLRAWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWAGKRPGVYTDYIYQGPMALVLLINFIFLFNIVRILMTKLRASTTSETIQARKAVKATLVLLPLLGITYMLAFVNPGEDEVSRVVFIYFNAFLESFQGFFVSVFACFLN