5j32 A 1.933 BS01 MG A 1 D288 D292 D258 D262 L48 Y181 K232 D264 D288 D292 L18 Y151 K202 D234 D258 D262 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 P93832 27137927 501 QMGRGSEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDS 5j32 A 1.933 BS02 IPM A 1 R136 R174 Y181 D288 R106 R144 Y151 D258 L48 Y181 K232 D264 D288 D292 L18 Y151 K202 D234 D258 D262 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 Kd=8.3uM -logKd/Ki=5.08, Kd=8.3uM P93832 27137927 502 QMGRGSEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDS 5j32 B 1.933 BS01 MG A 2 D288 D292 D253 D257 L48 Y181 K232 D264 D288 D292 L13 Y146 K197 D229 D253 D257 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 P93832 27137927 503 SEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDSQ 5j32 B 1.933 BS02 IPM A 2 R136 R146 R174 Y181 D288 R101 R111 R139 Y146 D253 L48 Y181 K232 D264 D288 D292 L13 Y146 K197 D229 D253 D257 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 -logKd/Ki=5.08, Kd=8.3uM P93832 27137927 504 SEFGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSVDSQ 5j32 C 1.933 BS01 MG C 1 D288 D292 D248 D252 L48 Y181 K232 D264 D288 D292 L8 Y141 K192 D224 D248 D252 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 P93832 27137927 501 KRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKS 5j32 C 1.933 BS02 IPM C 1 R136 R174 Y181 D288 R96 R134 Y141 D248 L48 Y181 K232 D264 D288 D292 L8 Y141 K192 D224 D248 D252 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 Kd=8.3uM P93832 27137927 502 KRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKS 5j32 D 1.933 BS01 MG C 2 D288 D292 D251 D255 L48 Y181 K232 D264 D288 D292 L11 Y144 K195 D227 D251 D255 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 P93832 27137927 503 FGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSV 5j32 D 1.933 BS02 IPM C 2 R136 R146 R174 Y181 D288 R99 R109 R137 Y144 D251 L48 Y181 K232 D264 D288 D292 L11 Y144 K195 D227 D251 D255 1.1.1.85 0000287,0003862,0005829,0008652,0009082,0009098,0009507,0009536,0009553,0009555,0009570,0009941,0016491,0016616,0042803,0046872,0051287,0070403 P93832 27137927 504 FGKKRYTITLLPGDGIGPEVVSIAKNVLQQAGSLEGVEFNFREMPIGGAALDLVGVPLPEETISAAKESDAVLLGAIGGYKWDNNEKHLRPEKGLLQIRAALKVFANLRPATVLPQLVDASTLKREVAEGVDLMVVRELTGGIYFGEPRGIKTNENGEEVGFNTEVYAAHEIDRIARVAFETARKRRGKLCSVDKANVLEASILWRKRVTALASEYPDVELSHMYVDNAAMQLVRDPKQFDTIVTNNIFGDILSDEASMITGSIGMLPSASLSDSGPGLFEPIHGSAPDIAGQDKANPLATILSAAMLLKYGLGEEKAAKRIEDAVLVALNNGFRTGDIYSAGTKLVGCKEMGEEVLKSV