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GPCR

NameGlucagon receptor
SpeciesMus musculus (Mouse)
GeneGcgr
SynonymGGR
GL-R
glucagon receptor
GR
DiseaseN/A for non-human GPCRs
Length485
Amino acid sequenceMPLTQLHCPHLLLLLLVLSCLPEAPSAQVMDFLFEKWKLYSDQCHHNLSLLPPPTELVCNRTFDKYSCWPDTPPNTTANISCPWYLPWYHKVQHRLVFKRCGPDGQWVRGPRGQPWRNASQCQLDDEEIEVQKGVAKMYSSQQVMYTVGYSLSLGALLLALVILLGLRKLHCTRNYIHGNLFASFVLKAGSVLVIDWLLKTRYSQKIGDDLSVSVWLSDGAMAGCRVATVIMQYGIIANYCWLLVEGVYLYSLLSLATFSERSFFSLYLGIGWGAPLLFVIPWVVVKCLFENVQCWTSNDNMGFWWILRIPVFLALLINFFIFVHIIHLLVAKLRAHQMHYADYKFRLARSTLTLIPLLGVHEVVFAFVTDEHAQGTLRSTKLFFDLFLSSFQGLLVAVLYCFLNKEVQAELMRRWRQWQEGKALQEERLASSHGSHMAPAGPCHGDPCEKLQLMSAGSSSGTGCVPSMETSLASSLPRLADSPT
UniProtQ61606
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL4773
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 39
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
311672D structureCHEMBL348555C24H22ClN3387.9112 / 26.1No
501452D structure643011-22-7C27H21ClF3N3O3S559.9889 / 26.4No
627412D structureCHEMBL350255C21H14BrClN2409.7111 / 15.9No
646462D structureMK 0893C32H27Cl2N3O4588.4855 / 26.8No
773492D structureCHEMBL347663C25H23ClN2O402.9222 / 16.5No
950772D structureCHEMBL158671C21H15FN2314.3632 / 14.7Yes
1147862D structureL-168,049C24H20BrClN2O467.7912 / 16.8No
1150162D structureaminothiazole, 10C30H27Cl2N3O3S580.5246 / 27.5No
1290122D structureglucagon receptor antagonists-4C26H28F3N3O4503.5228 / 25.0No
1324242D structureCHEMBL1644183C27H20Cl2F3N3O4578.3698 / 26.4No
1518722D structureCHEMBL328126C21H14ClFN2348.8052 / 15.3No
1744252D structureaminothiazole, 16C27H21ClF3N3O3S559.9889 / 26.4No
1793312D structureCHEMBL348401C21H21FN2320.4112 / 15.2No
1828872D structureCHEMBL155686C24H20Cl2N2O423.3372 / 16.7No
2028422D structureCHEMBL346698C23H19ClN2O374.8682 / 15.6No
2103522D structureCHEMBL158535C24H19ClN2O386.8792 / 15.8No
2167432D structureCHEMBL160561C24H21ClN2O388.8952 / 16.0No
2325702D structureCHEMBL351104C23H17ClN2O2388.8513 / 14.9Yes
2334182D structureCHEMBL158989C22H14FN3339.3733 / 14.4Yes
2384532D structureCHEMBL345834C27H27ClN2O430.9762 / 17.5No
2719262D structureCHEMBL156458C24H21ClN2O388.8952 / 16.1No
2860502D structureCHEMBL157529C21H14F2N2332.3543 / 14.8Yes
2895992D structureCHEMBL158676C25H23ClN2O402.9222 / 16.4No
3080652D structureCHEMBL347462C27H27ClN2O2446.9753 / 16.9No
3174012D structureCHEMBL160380C22H17ClN2O360.8412 / 15.2No
3242582D structureaminothiazole, 6C34H26F3N3O4S629.65410 / 27.7No
3249172D structureCHEMBL160638C21H13Cl2FN2383.2472 / 15.9No
3456802D structureCHEMBL160735C21H21ClN2336.8631 / 16.1No
3524942D structureaminothiazole, 19C28H21F6N3O4S609.54313 / 27.0No
3722602D structureaminothiazole, 7C30H26F3N3O3S565.6119 / 26.6No
3786332D structureCHEMBL158548C18H17ClN2296.7981 / 14.7Yes
3892052D structureCHEMBL160287C24H20BrClN2O467.7912 / 16.8No
3895452D structureaminothiazole, 17C27H21ClF3N3O4S575.98710 / 26.7No
3938692D structureCHEMBL155694C22H17ClN2O360.8412 / 15.2No
3981072D structureCHEMBL160372C15H11ClN2254.7171 / 13.6Yes
4011762D structureCHEMBL160490C21H14Cl2N2365.2571 / 15.8No
4152322D structureCHEMBL160281C21H14ClFN2348.8052 / 15.3No
4215252D structureCHEMBL345863C18H15ClN2O2326.783 / 13.8Yes
4232832D structureaminothiazole, 8C30H26F3N3O4S581.6110 / 26.9No

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