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GPCR

NameNeuropeptide Y receptor type 4
SpeciesRattus norvegicus (Rat)
GeneNpy4r
Synonymneuropeptide Y receptor type 4
NPY4-R
Pancreatic polypeptide receptor 1
PP1
Y4 receptor
DiseaseN/A for non-human GPCRs
Length375
Amino acid sequenceMNTSHLMASLSPAFLQGKNGTNPLDSLYNLSDGCQDSADLLAFIITTYSVETVLGVLGNLCLIFVTTRQKEKSNVTNLLIANLAFSDFLMCLICQPLTVTYTIMDYWIFGEVLCKMLTFIQCMSVTVSILSLVLVALERHQLIINPTGWKPSISQAYLGIVVIWFISCFLSLPFLANSILNDLFHYNHSKVVEFLEDKVVCFVSWSSDHHRLIYTTFLLLFQYCVPLAFILVCYMRIYQRLQRQRRAFHTHTCSSRVGQMKRINGMLMAMVTAFAVLWLPLHVFNTLEDWYQEAIPACHGNLIFLMCHLFAMASTCVNPFIYGFLNINFKKDIKALVLTCRCRPPQGEPEPLPLSTVHTDLSKGSMRMGSKSNVM
UniProtQ63447
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL4827
IUPHAR307
DrugBankN/A

Known ligands

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Total entries: 10
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
710892D structureNPY2-36, porcineC181H278N54O554090.5462 / 58-17.7No
934922D structureNPY D-Trp32C196H290N56O56S4358.8765 / 59-15.6No
1125132D structureCID 16142386C135H209N41O362982.4142 / 48-6.6No
1243632D structureBDBM82300C195H302N58O57S+44402.9761 / 65-14.8No
5547432D structure[125I]GW1229C110H170N34O242352.7848 / 386.8No
3248532D structurePP, BOVINEC186H291N53O54S2+24197.8159 / 56-12.3No
3438552D structureNucleopeptide YC190H287N55O574253.7164 / 63-15.5No
5552592D structurehuman Neuropeptide YC189H285N55O57S4271.7565 / 63-16.2No
4188622D structurePP,SALMONC185H289N53O54S2+24183.7859 / 56-12.7No
4393352D structureCHEMBL62166C27H24N4O3452.5144 / 23.4Yes

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