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You can:

Check the GPCR table for details.
Go to the ligand list to see ligands that interacts with this GPCR.
Go to the individual ligand page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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GPCR

Name	KiSS-1 receptor
Species	Rattus norvegicus (Rat)
Gene	Kiss1r
Synonym	Metastin receptor Kisspeptins receptor kisspeptin receptor KiSS1-derived peptide receptor KiSS-1R kiSS-1 receptor hOT7T175 GPR54 G-protein coupled receptor OT7T175 G-protein coupled receptor 54 rOT7T175 [ Show all ]
Disease	N/A for non-human GPCRs
Length	396
Amino acid sequence	MAAEATLGPNVSWWAPSNASGCPGCGVNASDGPGSAPRPLDAWLVPLFFAALMLLGLVGNSLVIFVICRHKHMQTVTNFYIANLAATDVTFLLCCVPFTALLYPLPTWVLGDFMCKFVNYIQQVSVQATCATLTAMSVDRWYVTVFPLRALHRRTPRLALTVSLSIWVGSAAVSAPVLALHRLSPGPHTYCSEAFPSRALERAFALYNLLALYLLPLLATCACYGAMLRHLGRAAVRPAPTDGALQGQLLAQRAGAVRTKVSRLVAAVVLLFAACWGPIQLFLVLQALGPSGAWHPRSYAAYALKIWAHCMSYSNSALNPLLYAFLGSHFRQAFCRVCPCGPQRQRRPHASAHSDRAAPHSVPHSRAAHPVRVRTPEPGNPVRRSPSVQDEHTAPL
UniProt	Q924U1
Protein Data Bank	N/A
GPCR-HGmod model	N/A
3D structure model	No available structures or models
BioLiP	N/A
Therapeutic Target Database	N/A
ChEMBL	CHEMBL1169599
IUPHAR	266
DrugBank	N/A

Known ligands

You can:

Click GLASS IDs to check the association information.
Click ligand names to check details of the ligands.
Download a TSV version of all interaction information.
Download a SDF structure collection of all known ligands.

GLASS ID	Molecule	Formula	Molecular weight	H-bond acceptor / donor	XlogP	Lipinski's druglikeness
514	CHEMBL3085807	C60H88N18O13	1269.48	16 / 17	-1.1	No
441716	CHEMBL3314214	C60H79N17O12	1230.4	15 / 16	-0.3	No
536076	CHEMBL3928465	C64H82FN17O13	1316.46	15 / 18	1.3	No
548025	CHEMBL3982675	C59H82N16O13	1223.4	14 / 16	-0.3	No
442502	CHEMBL3314224	C64H83N17O13	1298.47	14 / 18	1.2	No
548125	CHEMBL3985112	C64H83N17O13	1298.47	14 / 18	1.2	No
536712	CHEMBL3977314	C58H79FN16O15	1259.36	17 / 18	-1.0	No
442826	CHEMBL3314227	C69H85N17O13	1360.55	14 / 19	3.1	No
36835	CHEMBL2151645	C64H85N17O14	1316.49	16 / 18	-1.2	No
536953	CHEMBL3939287	C55H75FN16O13	1187.3	15 / 17	-0.9	No
536983	CHEMBL3985323	C56H78N16O13	1183.34	14 / 17	-1.1	No
40351	CHEMBL3087930	C56H81N17O15	1232.37	17 / 19	-3.8	No
40354	CHEMBL2151648	C56H81N17O15	1232.37	17 / 19	-3.8	No
537090	CHEMBL3931718	C57H78N16O13	1195.35	14 / 16	-1.1	No
443575	CHEMBL3314225	C66H87N17O13	1326.53	14 / 18	2.0	No
62322	CHEMBL2151651	C60H82N18O14	1279.43	17 / 18	-2.6	No
444447	CHEMBL3314217	C63H83N17O11	1254.46	13 / 17	2.5	No
444602	CHEMBL3314209	C60H81N17O11	1216.42	14 / 16	1.3	No
548938	CHEMBL3964403	C63H82N16O13	1271.45	14 / 16	0.8	No
548989	CHEMBL3976038	C59H84N16O13	1225.42	14 / 17	0.8	No
445502	CHEMBL3314221	C61H80N16O11	1213.41	13 / 17	2.4	No
445523	CHEMBL3314220	C60H78N16O11	1199.39	13 / 17	2.0	No
445635	CHEMBL3314218	C57H76N16O11	1161.34	14 / 16	0.8	No
445748	CHEMBL3314219	C58H78N16O12	1191.36	15 / 17	0.2	No
103484	CHEMBL2151646	C63H84N18O14	1317.48	16 / 19	-1.4	No
103486	CHEMBL2151654	C63H84N18O14	1317.48	16 / 19	-1.4	No
103488	CHEMBL3085804	C63H84N18O14	1317.48	16 / 19	-1.4	No
103489	CHEMBL3087925	C63H84N18O14	1317.48	16 / 19	-1.4	No
561238	CHEMBL1171977	C27H22FN5O4	499.502	8 / 3	4.0	Yes
133224	CHEMBL3086282	C61H79N15O12	1214.4	14 / 16	1.5	No
147150	CHEMBL2151647	C55H79N17O15	1218.34	17 / 19	-4.2	No
539771	CHEMBL3956072	C57H78N16O13S	1227.41	15 / 16	-0.2	No
561974	CHEMBL1173008	C29H26FN5O3	511.557	8 / 2	5.0	No
539918	CHEMBL3967058	C57H78N16O13	1195.35	14 / 16	-0.6	No
158936	CHEMBL3085810	C51H73N15O13	1104.24	15 / 17	-2.4	No
540147	CHEMBL3915251	C56H78N16O13	1183.34	14 / 17	-0.6	No
549937	CHEMBL3904889	C56H78N16O13	1183.34	14 / 17	-0.6	No
540214	CHEMBL3964945	C57H80N16O13	1197.37	14 / 17	-0.4	No
448232	CHEMBL3314216	C62H81N17O12	1256.44	14 / 18	0.9	No
167307	CHEMBL3085805	C57H80N18O13	1225.38	15 / 18	-2.7	No
540376	CHEMBL3894943	C59H82N16O13	1223.4	14 / 16	0.1	No
448491	CHEMBL3314212	C66H82N18O11	1303.5	14 / 18	2.4	No
174046	CHEMBL3087793	C62H82N18O14	1303.45	16 / 19	-1.9	No
176245	CHEMBL3086281	C57H77N15O12	1164.34	14 / 16	0.2	No
178500	CHEMBL3087926	C62H83N17O14	1290.45	16 / 19	-1.0	No
563096	CHEMBL1169902	C28H24FN5O4	513.529	8 / 3	3.9	No
541000	CHEMBL3938759	C60H78N16O13	1231.38	14 / 17	1.1	No
449424	CHEMBL3315315	C65H84N18O14	1341.5	16 / 20	-1.4	No
201328	CHEMBL2151649	C58H85N17O14	1244.42	16 / 18	-1.8	No
541657	UNII-YO029HR229	C58H80N16O14	1225.38	15 / 17	-1.2	No
217834	CHEMBL3085809	C59H78N16O12	1203.37	14 / 17	0.3	No
217836	CHEMBL3086283	C59H78N16O12	1203.37	14 / 17	0.3	No
550599	CHEMBL3911692	C58H80N16O13	1209.38	14 / 16	-0.3	No
550600	CHEMBL3966187	C58H80N16O13	1209.38	14 / 16	-0.3	No
542107	CHEMBL3958495	C58H80N16O15	1241.38	16 / 18	-1.1	No
550757	CHEMBL3984058	C58H80N16O15	1241.38	16 / 18	-1.1	No
237411	CHEMBL2151644	C64H87N17O13	1302.51	16 / 18	-1.2	No
451492	CHEMBL3314228	C61H81N17O13	1260.43	15 / 17	0.0	No
451520	CHEMBL3314207	C58H77N17O12	1204.36	15 / 17	-0.7	No
451836	CHEMBL3314213	C60H79N17O11	1214.4	14 / 15	0.6	No
265525	CHEMBL3086280	C54H79N15O12	1130.32	14 / 16	-0.1	No
543087	CHEMBL3949224	C59H84FN17O13	1258.43	16 / 18	-0.7	No
271174	CHEMBL2151643	C64H85N17O13S	1332.55	16 / 18	-0.8	No
543346	CHEMBL3956626	C56H78N16O13	1183.34	14 / 16	-0.8	No
281556	CID 72711590	C65H85N19O13	1340.52	16 / 20	0.2	No
452800	CHEMBL3314210	C63H79N17O11	1250.43	14 / 16	1.6	No
285672	CHEMBL3085811	C52H75N15O13	1118.26	15 / 17	-2.0	No
297196	Kisspeptin-10	C63H83N17O14	1302.46	16 / 18	-1.9	No
544069	CHEMBL3949159	C64H82FN17O13	1316.46	15 / 18	1.3	No
544071	CHEMBL3930297	C64H82FN17O13	1316.46	15 / 18	1.3	No
453661	CHEMBL3314226	C66H85N17O13	1324.51	14 / 18	1.6	No
566795	CHEMBL1170903	C29H24FN5O4	525.54	8 / 4	4.0	No
566797	CHEMBL1170904	C29H24FN5O4	525.54	8 / 4	4.0	No
544584	CHEMBL3921327	C64H82ClN17O13	1332.92	14 / 18	1.8	No
551906	CHEMBL3957784	C64H82FN17O13	1316.46	15 / 18	1.3	No
324484	CHEMBL3085806	C62H83N19O13	1302.47	16 / 18	-2.1	No
567738	CHEMBL1173643	C27H22FN5O3	483.503	8 / 3	4.2	Yes
338066	CHEMBL3086285	C56H76N16O11	1149.32	14 / 15	-0.5	No
455266	CHEMBL3314211	C61H83N17O11	1230.44	14 / 16	1.7	No
552246	CHEMBL3914238	C59H85N17O13	1240.44	15 / 18	-0.8	No
545361	CHEMBL3956437	C59H85N17O13	1240.44	15 / 18	-0.8	No
545392	CHEMBL3977235	C57H80N16O13	1197.37	14 / 16	-0.4	No
545395	CHEMBL3947975	C57H80N16O13	1197.37	14 / 16	-0.4	No
455687	CHEMBL3314208	C59H79N17O12	1218.39	15 / 17	-0.3	No
545804	CHEMBL3968824	C57H79FN16O13	1215.36	15 / 17	-0.3	No
368145	CHEMBL2151653	C65H85N17O14	1328.5	16 / 18	-0.3	No
377629	CHEMBL3087929	C61H89N17O14	1284.49	16 / 18	-0.4	No
377631	CHEMBL2151650	C61H89N17O14	1284.49	16 / 18	-0.4	No
457343	CHEMBL3314223	C62H80N16O12	1241.42	13 / 17	1.7	No
393559	CHEMBL3086286	C58H77N17O11	1188.36	14 / 16	-0.4	No
400268	CHEMBL3087928	C61H83N17O14	1278.44	16 / 18	-1.6	No
457839	CHEMBL3314229	C62H82N16O13	1259.44	14 / 17	1.0	No
547066	CHEMBL3896533	C55H76N16O13	1169.31	14 / 17	-1.0	No
547112	CHEMBL3967782	C58H79FN16O14	1243.37	16 / 17	-1.1	No
418463	CHEMBL3086284	C56H76N16O12	1165.32	15 / 16	-0.9	No
423400	CHEMBL2151642	C64H85N17O14	1316.49	16 / 18	-1.4	No
458540	CHEMBL3314215	C61H79N17O12	1242.41	14 / 18	0.5	No
570527	CHEMBL1169901	C27H22FN5O4	499.502	8 / 4	4.0	Yes
427583	CHEMBL3087931	C60H82N18O14	1279.43	17 / 18	-2.6	No
427584	CHEMBL2151652	C60H82N18O14	1279.43	17 / 18	-2.6	No