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GPCR-RD is a database for experimental restaints of GPCRs. Although no solved X-ray or NMR structure is available for most GPCR sequences, numerous experiments have been performed on GPCRs to identify the critical residues and motifs. Experimental restraints were systematically collected from the literature using an automated text mining algorithm combined with manual validation, with the purpose of assisting GPCR 3-D structure modeling and function annotation. The GPCR-RD data are useful for GPCR 3D structure modeling, such as the GPCR-I-TASSER algorithm. The flow chart below summarizes the procedure for the extraction of experimental data and spatial restraints from literature and other resources.

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11002 entries in GPCR-RD.
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GPCR-RD: GPCR experimental restaint database
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Swiss-Prot ID Experimental Data Swiss-Prot ID Experimental Data Swiss-Prot ID Experimental Data
opsd_bovin R147Q opsd_bovin F148A opsd_bovin G149A
opsd_bovin H152N opsd_bovin S176F opsd_bovin E181A
opsd_bovin E181C opsd_bovin E181D opsd_bovin E181F
opsd_bovin E181G opsd_bovin E181H opsd_bovin E181I
opsd_bovin E181K opsd_bovin E181L opsd_bovin E181M
opsd_bovin E181N opsd_bovin E181P opsd_bovin E181Q
opsd_bovin E181R opsd_bovin E181S opsd_bovin E181T
opsd_bovin E181V opsd_bovin E181W opsd_bovin E181Y
opsd_bovin C185 opsd_bovin S186A opsd_bovin S186D
opsd_bovin S186I opsd_bovin C187 opsd_bovin G188R
opsd_bovin G188S opsd_bovin T198C opsd_bovin N200C
opsd_bovin Q225C opsd_bovin V227C opsd_bovin A233G
opsd_bovin A233N opsd_bovin A234G opsd_bovin A234N
opsd_bovin A235G opsd_bovin A235N opsd_bovin S240A
opsd_bovin T242A opsd_bovin T243A opsd_bovin T243V
opsd_bovin E247C opsd_bovin K248C opsd_bovin K248L
opsd_bovin E249C opsd_bovin V250A opsd_bovin V250C
opsd_bovin T251A opsd_bovin T251C opsd_bovin T251H
opsd_bovin R252A opsd_bovin R252C opsd_bovin T277A
opsd_bovin F313A opsd_bovin F313C opsd_bovin C316
opsd_bovin C316S opsd_bovin C322 opsd_bovin C322S
opsd_bovin C323 opsd_bovin C323S opsd_bovin S334A
opsd_bovin T335A opsd_bovin T336A opsd_bovin T336P
opsd_bovin S338A opsd_bovin T340A opsd_bovin T340E
opsd_bovin T342A opsd_bovin S343A opsd_bovin S343E
opsd_canfa T4K opsd_canfa T4R opsd_mouse C322T
opsd_mouse C323S opsd_mouse E341X opsd_mouse Q344X
opsd_mouse V345M opsd_mouse P347L opsd_rat P23H
opsd_rat S281A opsd_ranpi Electron Microscopy 7 TMhelix x-y coordinates 6.99 14.20 12.73 24.69 20.70 22.08 28.55 23.88 28.98 13.10 21.47 7.47 14.62 12.96  [Electron Microscopy] opsd_todpa Electron Microscopy 7 TMhelix x-y coordinates 11.70 11.87 9.23 23.60 16.20 29.93 24.28 25.92 32.14 22.36 25.86 16.13 18.89 16.97  [Electron Microscopy]
opsx_human I49A  [Orientation Restraint] opsx_human T213I ptafr_cavpo S305G
ptafr_cavpo T335A pd2r_mouse A19P pd2r_mouse G22S


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