You can:

Go to the GPCR, ligand, or experimental data tables.
Go to the experimental data table for text mining information in PubMed ID column.
Go to the GPCR page and check other ligands which interact with it.
Go to the ligand page and check other GPCRs which it interacts with.
Go back to previous page.

GPCR

Name	Delta-type opioid receptor
Species	Homo sapiens (Human)
Gene	OPRD1
Synonym	D-OR-1 DOR opioid receptor OP1 DOP DOPr DOR-1 Delta receptor [ Show all ]
Disease	Cough Overactive bladder disorder Bladder disease Moderate-to-severe pain Diarrhea-predominant IBS Major depressive disorder Urinary incontinence Rheumatoid arthritis Premature ejaculation Pain Acute migraine Ischemic heart diseases Acute nonspecific diarrhea; Chronic diarrhea associated with inflammatory bowel disease Alcohol use disorders Anxiety disorder [ Show all ]
Length	372
Amino acid sequence	MEPAPSAGAELQPPLFANASDAYPSACPSAGANASGPPGARSASSLALAIAITALYSAVCAVGLLGNVLVMFGIVRYTKMKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELLCKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVGVPIMVMAVTRPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRLRSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDIDRRDPLVVAALHLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRKPCGRPDPSSFSRAREATARERVTACTPSDGPGGGAAA
UniProt	P41143
Protein Data Bank	4rwd, 4rwa, 4n6h
GPCR-HGmod model	P41143
3D structure model	This structure is from PDB ID 4rwd.
BioLiP	BL0303696,BL0303697, BL0265712, BL0265705,BL0265706,BL0265707,, BL0303699,BL0303701, BL0303698,BL0303700
Therapeutic Target Database	T58992
ChEMBL	CHEMBL236
IUPHAR	317
DrugBank	BE0000420

Ligand

Name	AC1MHY5M
Molecular formula	C26H26N2O3
IUPAC name	(21S)-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.01,13.02,21.04,12.05,10.019,25]pentacosa-4(12),5,7,9,15,17,19(25)-heptaene-2,16-diol
Molecular weight	414.505
Hydrogen bond acceptor	4
Hydrogen bond donor	3
XlogP	3.3
Synonyms	(21R)-22-(cyclopropylmethyl)-14-oxa-11,22-diazaheptacyclo[13.9.1.0^{1,13}.0^{2,21}.0^{4,12}.0^{5,10}.0^{19,25}]pentacosa-4(12),5,7,9,15,17,19(25)-heptaene-2,16-diol (8R)-7-(cyclopropylmethyl)-5,6,7,8,14,14b-hexahydro-4,8-methano[1]benzofuro[2,3-a]pyrido[4,3-b]carbazole-1,8a(9H)-diol BDBM21864
Inchi Key	WIYUZYBFCWCCQJ-XEWUMVRVSA-N
Inchi ID	InChI=1S/C26H26N2O3/c29-19-8-7-15-11-20-26(30)12-17-16-3-1-2-4-18(16)27-22(17)24-25(26,21(15)23(19)31-24)9-10-28(20)13-14-5-6-14/h1-4,7-8,14,20,24,27,29-30H,5-6,9-13H2/t20-,24?,25?,26?/m0/s1
PubChem CID	3034754
ChEMBL	N/A
IUPHAR	N/A
BindingDB	21864
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand satisfies Lipinski's rule of five.

Parameter	Value	Reference	Database source
EC50	0.11 nM	PMID12825957, PMID12672258	BindingDB
IC50	0.32 nM	PMID1335078	BindingDB
IC50	0.39 nM	PMID19282177	BindingDB
Ki	0.02 nM	PMID8114680	BindingDB
Ki	0.03 nM	PMID1333013	BindingDB
Ki	0.03 nM	PMID7853332, PMID2160538	BindingDB
Ki	0.031 nM	PMID1648136	BindingDB
Ki	0.04 nM	PMID12565965	BindingDB
Ki	0.062 nM	PMID14998329, PMID12431065, PMID10229636	BindingDB
Ki	0.07 nM	PMID14711299	BindingDB
Ki	0.14 nM	PMID19282177	BindingDB
Ki	0.15 nM	PMID11294396	BindingDB
Ki	0.16 nM	PMID12930147	BindingDB
Ki	0.2 nM	PMID15588100, PMID12672258, PMID15456250, PMID11784158, PMID12825957	BindingDB
Ki	0.2 nM	PMID9686407	BindingDB
Ki	0.22 nM	PMID11597422	BindingDB
Ki	0.24 nM	PMID12930147	BindingDB
Ki	0.46 nM	PMID21621410	BindingDB
Ki	0.5 nM	PMID21621410	BindingDB
Ki	1.04 nM	PMID7932177	BindingDB
Ki	2.0 nM	PMID19595591	BindingDB