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GPCR

NameGlucagon-like peptide 1 receptor
SpeciesRattus norvegicus (Rat)
GeneGlp1r
SynonymGLP-1 receptor
GLP-1-R
GLP-1R
glucagon-like peptide 1 receptor
DiseaseN/A for non-human GPCRs
Length463
Amino acid sequenceMAVTPSLLRLALLLLGAVGRAGPRPQGATVSLSETVQKWREYRHQCQRFLTEAPLLATGLFCNRTFDDYACWPDGPPGSFVNVSCPWYLPWASSVLQGHVYRFCTAEGIWLHKDNSSLPWRDLSECEESKQGERNSPEEQLLSLYIIYTVGYALSFSALVIASAILVSFRHLHCTRNYIHLNLFASFILRALSVFIKDAALKWMYSTAAQQHQWDGLLSYQDSLGCRLVFLLMQYCVAANYYWLLVEGVYLYTLLAFSVFSEQRIFKLYLSIGWGVPLLFVIPWGIVKYLYEDEGCWTRNSNMNYWLIIRLPILFAIGVNFLVFIRVICIVIAKLKANLMCKTDIKCRLAKSTLTLIPLLGTHEVIFAFVMDEHARGTLRFVKLFTELSFTSFQGFMVAVLYCFVNNEVQMEFRKSWERWRLERLNIQRDSSMKPLKCPTSSVSSGATVGSSVYAATCQNSCS
UniProtP32301
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL5862
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 12
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
929342D structureCID 46883767C208H319N49O63S4546.1868 / 58-11.4No
1228042D structureCID 46883764C232H357N49O69S4968.7473 / 63-7.8No
1237372D structureBDBM50241203C184H282N50O60S4186.6366 / 57-21.3No
1561942D structureCID 46883763C208H319N49O65S4578.1870 / 60-14.1No
1588632D structureCHEMBL449327C54H52N4O16S21077.1418 / 68.3No
1834162D structureCHEMBL2158415C28H28N2O8S552.5989 / 34.5No
2212002D structureCHEMBL510593C56H52N4O14S21069.1716 / 68.6No
2533932D structureCID 46883762C208H319N49O65S4578.1870 / 60-14.1No
2680392D structureBDBM50314042C232H357N49O65S4904.7569 / 58-2.8No
3391592D structureGLP-1 (1-37) amideC186H275N51O594169.5466 / 63-17.1No
4113772D structureBDBM50314039C208H319N49O64S4562.1869 / 58-13.1No
4206282D structureBDBM50314040C232H357N49O67S4936.7471 / 60-5.4No

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