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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameMuscarinic acetylcholine receptor M4
SpeciesBos taurus (Bovine)
GeneCHRM4
SynonymN/A
DiseaseN/A for non-human GPCRs
Length126
Amino acid sequenceMKQSVKKPPPPGDTTVRGELPNGKLEEAPPPVLPPPPRPMADKDTSNESSSGSATQNTKERPPTELSTTEATTPATPAPPLQPRTLNPASKWSKIQIVTKQTGNECVTAIEIVPATPAGMRPAANV
UniProtP41986
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLN/A
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 9
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
228752D structuretropicamideC17H20N2O2284.3593 / 11.5Yes
821612D structureAC1L1AYEC22H35NO2345.5273 / 05.0Yes
1270992D structure4-Diphenylacetoxy-1,1-dimethylpiperidiniumC21H26NO2+324.4442 / 04.0Yes
2862132D structurehexahydrosiladifenidolC20H33NOSi331.5752 / 1N/AN/A
2997402D structurepirenzepineC19H21N5O2351.415 / 10.1Yes
3020062D structureMethoctramineC36H62N4O2582.9186 / 46.8No
3226252D structurescopolamineC17H21NO4303.3585 / 10.9Yes
3634532D structureTelenzepineC19H22N4O2S370.4715 / 11.7Yes
4195412D structureTripitramineC64H77N13O61124.4113 / 47.7No

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