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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

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GPCR

NameGastric inhibitory polypeptide receptor
SpeciesRattus norvegicus (Rat)
GeneGipr
SynonymGIP receptor
GIP-R
Gippr
Glucose-dependent insulinotropic polypeptide receptor
DiseaseN/A for non-human GPCRs
Length455
Amino acid sequenceMPLRLLLLLLWLWGLSLQRAETDSEGQTTGELYQRWERYGWECQNTLEATEPPSGLACNGSFDMYACWNYTAANTTARVSCPWYLPWYRQVAAGFVFRQCGSDGQWGSWRDHTQCENPEKNGAFQDQKLILERLQVVYTVGYSLSLATLLLALLILSLFRRLHCTRNYIHMNLFTSFMLRAGAILTRDQLLPPLGPYTGNQTPTLWNQALAACRTAQILTQYCVGANYTWLLVEGVYLHHLLVVVRRSEKGHFRCYLLLGWGAPALFVIPWVIVRYLYENTQCWERNEVKAIWWIIRTPILITILINFLIFIRILGILVSKLRTRQMRCPDYRLRLARSTLTLMPLLGVHEVVFAPVTEEQAEGSLRFAKLAFEIFLSSFQGFLVSVLYCFINKEVQSEIRRLRLSLQEQCPRPHLGQAPRAVPLSSAPQEAAIRNALPSGMLHVPGDEVLESYC
UniProtP43219
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL5001
IUPHARN/A
DrugBankN/A

Known ligands

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Total entries: 4
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
369062D structureGRA EX-25C29H36F3N3O5563.6188 / 35.8No
441902D structureCipargaminC19H14Cl2FN3O390.2393 / 33.9Yes
3555792D structureCHEMBL386446C30H29Cl2N3O4566.4794 / 35.9No
3966222D structureCHEMBL487476C30H29Cl2N3O5582.4785 / 45.4No

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