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GPCR

NameNeuromedin-K receptor
SpeciesMus musculus (Mouse)
GeneTacr3
SynonymTac3r
SP-N receptor
Nmkr
NKR
NK3 receptor
[ Show all ]
DiseaseN/A for non-human GPCRs
Length452
Amino acid sequenceMASVPTGENWTDGTAGVGSHTGNLSAALGITEWLALQAGNFSSALGLPVTSQAPSQVRANLTNQFVQPSWRIALWSLAYGLVVAVAVFGNLIVIWIILAHKRMRTVTNYFLVNLAFSDASVAAFNTLVNFIYGVHSEWYFGANYCRFQNFFPITAVFASIYSMTAIAVDRYMAIIDPLKPRLSATATKIVIGSIWILAFLLAFPQCLYSKIKVMPGRTLCYVQWPEGPKQHFTYHIIVIILVYCFPLLIMGVTYTIVGITLWGGEIPGDTCDKYHEQLKAKRKVVKMMIIVVVTFAICWLPYHVYFILTAIYQQLNRWKYIQQVYLASFWLAMSSTMYNPIIYCCLNKRFRAGFKRAFRWCPFIQVSSYDELELKTTRFHPTRQSSLYTVSRMESVTVLYDPSEGDPAKSSRKKRAVPRDPSANGCSHREFKSASTTSSFISSPYTSVDEYS
UniProtP47937
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLN/A
IUPHAR362
DrugBankN/A

Known ligands

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Total entries: 14
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
5532582D structureSubstance PC63H98N18O13S1347.6517 / 15-2.3No
4598862D structureCHEMBL299377C35H41Cl2N3O2606.6323 / 07.0No
5538192D structureNEUROKININ AC50H80N14O14S1133.3318 / 16-4.8No
5538702D structureSenktideC40H55N7O11S841.97812 / 81.1No
4608672D structureNKB [MePhe7]C56H81N13O14S21224.4618 / 13-1.4No
4610602D structureGR 113808C19H27N3O4S393.5026 / 11.7Yes
5543832D structureNeurokinin BC55H79N13O14S21210.4318 / 14-1.6No
4615102D structurevenlafaxineC17H27NO2277.4083 / 12.9Yes
4617642D structureSB 235375C27H24N2O4440.4995 / 25.1No
4617942D structureBCTCC20H25ClN4O372.8973 / 14.3Yes
4618162D structureabt-702C22H19BrN6O463.3397 / 13.4Yes
4622772D structureN-Methyl-3-phenyl-3-(o-tolyloxy)propan-1-amineC17H21NO255.3612 / 13.7Yes
4628362D structureduloxetineC18H19NOS297.4163 / 14.3Yes
4628872D structureBurapitantC31H35Cl2F6N3O3682.52910 / 16.2No

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