Home Research COVID-19 Services Publications People Teaching Job Opening News Forum Lab Only
Online Services

I-TASSER I-TASSER-MTD C-I-TASSER CR-I-TASSER QUARK C-QUARK LOMETS MUSTER CEthreader SEGMER DeepFold DeepFoldRNA FoldDesign COFACTOR COACH MetaGO TripletGO IonCom FG-MD ModRefiner REMO DEMO DEMO-EM DMFold SPRING COTH Threpp PEPPI BSpred ANGLOR EDock BSP-SLIM SAXSTER FUpred ThreaDom ThreaDomEx EvoDesign BindProf BindProfX SSIPe GPCR-I-TASSER MAGELLAN ResQ STRUM DAMpred

TM-score TM-align US-align MM-align RNA-align NW-align LS-align EDTSurf MVP MVP-Fit SPICKER HAAD PSSpred 3DRobot MR-REX I-TASSER-MR SVMSEQ NeBcon ResPRE TripletRes DeepPotential WDL-RF ATPbind DockRMSD DeepMSA FASPR EM-Refiner GPU-I-TASSER

BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP Tara-3D TM-fold DECOYS POTENTIAL RW/RWplus EvoEF HPSF THE-DB ADDRESS Alpaca-Antibody CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13 CASP14

You can:

GPCR

NameUracil nucleotide/cysteinyl leukotriene receptor
SpeciesHomo sapiens (Human)
GeneGPR17
SynonymGPR17
P2Y-like receptor
G-protein coupled receptor 17
R12
UDP/CysLT receptor
[ Show all ]
DiseaseN/A
Length367
Amino acid sequenceMSKRSWWAGSRKPPREMLKLSGSDSSQSMNGLEVAPPGLITNFSLATAEQCGQETPLENMLFASFYLLDFILALVGNTLALWLFIRDHKSGTPANVFLMHLAVADLSCVLVLPTRLVYHFSGNHWPFGEIACRLTGFLFYLNMYASIYFLTCISADRFLAIVHPVKSLKLRRPLYAHLACAFLWVVVAVAMAPLLVSPQTVQTNHTVVCLQLYREKASHHALVSLAVAFTFPFITTVTCYLLIIRSLRQGLRVEKRLKTKAVRMIAIVLAIFLVCFVPYHVNRSVYVLHYRSHGASCATQRILALANRITSCLTSLNGALDPIMYFFVAEKFRHALCNLLCGKRLKGPPPSFEGKTNESSLSAKSEL
UniProtQ13304
Protein Data BankN/A
GPCR-HGmod modelQ13304
3D structure modelThis predicted structure model is from GPCR-EXP Q13304.
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL1075162
IUPHAR88
DrugBankN/A

Known ligands

You can:

Total entries: 51
Page:  / 1 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
388172D structureCHEMBL129841C11H17N5O9P2425.23113 / 5-2.9No
470652D structureCID 11954340C17H21Cl2F3N5Na4O12P3S2864.27421 / 3N/ANo
496682D structureSCHEMBL9186131C12H10BrNO4312.1194 / 32.4Yes
715292D structureCHEMBL1098419C12H18ClN4O13P3554.66216 / 7-3.8No
752242D structureCHEMBL1094760C10H14ClN5O9P2445.64613 / 5-2.0No
918412D structure2'-Deoxy-N6-methyl adenosine 3',5'-diphosphate diammonium saltC11H23N7O9P2459.29313 / 5N/ANo
5383212D structureCHEMBL3968577C18H15NO4309.3214 / 33.3Yes
948462D structureUridine-5'-diphosphate sodium salt(1:3)C9H11N2Na3O12P2470.10612 / 3N/ANo
5537852D structureleukotriene C4C30H47N3O9S625.77811 / 70.7No
5538592D structureASN 04885796C28H28FN5O4517.5617 / 13.8No
1182102D structureCHEMBL1096742C15H36N9O13P3643.42421 / 11N/ANo
5538972D structureUdp galactoseC15H24N2O17P2566.30217 / 9-6.3No
5538992D structureUDP-glucoseC15H24N2O17P2566.30217 / 9-6.3No
1449342D structureSCHEMBL9186177C12H10BrNO4312.1194 / 32.4Yes
5399012D structureCHEMBL53914C12H9F2NO4269.2046 / 31.9Yes
5540302D structureASN 04421891C30H32N6O3524.6257 / 13.8No
5541262D structureASN 02563583C25H24N4O3S460.5526 / 14.8Yes
1732342D structureMdl-29951C12H9Cl2NO4302.1074 / 32.9Yes
1732352D structureCHEMBL3264006C12H9Cl2NO4310.1394 / 32.9Yes
1841862D structureCHEMBL1094109C11H18N5O13P3521.20817 / 7-5.0No
5409522D structureCHEMBL3897541C14H15NO4261.2774 / 32.4Yes
2158902D structureCHEMBL3132880C12H9Br2NO4391.0154 / 33.0Yes
2193902D structurePranlukastC27H23N5O4481.5127 / 24.2Yes
2295942D structureCHEMBL1097652C18H20N5O13P3607.30117 / 7-3.7No
2375942D structureCHEMBL3132881C12H9I2NO4485.0164 / 33.0Yes
2464132D structureCHEMBL1094760C10H20ClN7O9P2479.70815 / 7N/ANo
2542572D structureCHEMBL3132886C12H10INO4359.1194 / 32.3Yes
2546402D structureCHEMBL1097279C17H21Cl2F3N5O12P3S2-4772.31421 / 3-1.3No
2739272D structureCHEMBL3132882C14H9F6NO4369.21910 / 33.4Yes
2754122D structureCHEMBL50976C14H15NO6293.2756 / 31.6Yes
2888292D structureCHEMBL1094109C11H30N9O13P3589.33221 / 11N/ANo
3026042D structureCHEMBL1094759C9H22IN5O12P2581.1515 / 9N/ANo
3071822D structureCHEMBL1096742C15H24N5O13P3575.317 / 7-3.8No
5672242D structureASN 06917370C24H21ClF3N7O2531.9248 / 23.6No
5446612D structureCHEMBL3915176C24H19NO4385.4194 / 34.9Yes
3274452D structureCHEMBL590494C9H13IN2O12P2530.05712 / 6-4.4No
5549032D structureASN 04450772C26H25N5O6S535.5759 / 42.6No
3333052D structuremontelukastC35H36ClNO3S586.1875 / 27.7No
3366312D structureCHEMBL3132883C12H8Cl2FNO4320.0975 / 33.0Yes
3651682D structureCHEMBL1098419C12H30ClN8O13P3622.78620 / 11N/ANo
3823822D structureCHEMBL1098083C11H29ClN9O13P3623.77421 / 11N/ANo
3859702D structureGavestinelC18H12Cl2N2O3375.2053 / 34.4Yes
3860452D structureCHEMBL1097652C18H32N9O13P3675.42521 / 11N/ANo
3881352D structureuridine-5'-diphosphateC9H11N2O12P2-3401.13712 / 3-5.0No
5552432D structureUridine 5'-diphosphateC9H14N2O12P2404.16112 / 6-4.7No
3956042D structureCHEMBL3132887C12H10INO4359.1194 / 32.3Yes
5553182D structureleukotriene D4C25H40N2O6S496.6638 / 51.4Yes
5471092D structureCHEMBL3921330C15H13Cl2NO6374.176 / 32.3Yes
5473412D structure3-(2-carboxyethyl)-6-chloro-1H-indole-2-carboxylic AcidC12H10ClNO4267.6654 / 32.3Yes
5554262D structureAdenosine triphosphateC10H16N5O13P3507.18117 / 7-5.7No
4382512D structureCHEMBL1098083C11H17ClN5O13P3555.6517 / 7-4.1No

zhanglabzhanggroup.org | (734) 647-1549 | 100 Washtenaw Avenue, Ann Arbor, MI 48109-2218