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Check the ligand table for details.
Go to the GPCR list to see GPCRs with which this ligand interacts.
Go to the individual GPCR page for PubMed ID information by text mining.
Download a TSV version of all interaction data.
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Ligand

Name	Amentoflavone
Molecular formula	C30H18O10
IUPAC name	8-[5-(5,7-dihydroxy-4-oxochromen-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)chromen-4-one
Molecular weight	538.464
Hydrogen bond acceptor	10
Hydrogen bond donor	6
XlogP	5.0
Synonyms	1617-53-4 5,5',7,7'-Tetrahydroxy-2,2'-bis(4-hydroxyphenyl)-[3,8'-bi-4H-1-benzopyran]-4,4'-dione 8-[5-(5,7-dihydroxy-4-oxochromen-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)chromen-4-one. Amentoflavone, >=99.0% (HPLC) CHEBI:2631 HMS2228B12 MFCD20275041 Q-100192 UNII-9I1VC79L77 4',4''',5,5'',7,7''-Hexahydroxy-3''',8-biflavone, 8CI 8-(5-(5,7-dihydroxy-4-oxo-4H-chromen-2-yl)-2 A810291 BCP13255 CTK8F7701 I07-0160 N2268 SMR000156235 ZINC3984030 4H-1-Benzopyran-4-one, 8-[5-(5,7-dihydroxy-4-oxo-4H-1-benzopyran-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl) 8-[5-(5,7-dihydroxy-4-oxo-chromen-2-yl)-2-hydroxy-phenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)chromen-4-one Amenthoflavone C10018 DTXSID20167225 MEGxp0_000924 NSC-295677 SR-01000721725-3 (4-hydroxyphenyl)-4H-chromen-4-one 3',8''-Biapigenin 617A534 8-[5-[5,7-bis(oxidanyl)-4-oxidanylidene-chromen-2-yl]-2-oxidanyl-phenyl]-2-(4-hydroxyphenyl)-5,7-bis(oxidanyl)chromen-4-one Amentoflavone, analytical standard HMS3343J17 MLS000574827 SC-13592 W1536 4',5,7-Trihydroxyflavone(3'->8)-4',5,7-trihydroxyflavone 8-[5-(5,7-dihydroxy-4-oxo-1-benzopyran-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)-1-benzopyran-4-one AC1NQYPA BIDD:PXR0028 D06HRX KS-00000037 NCGC00247542-01 SR-01000721725 4H-1-Benzopyran-4-one,8-[5-(5,7-dihydroxy-4-oxo-4H-1-benzopyran-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)- 8-[5-(5,7-dihydroxy-4-oxochromen-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)chromen-4-one CC-24050 FT-0622262 MFCD00017470 NSC295677 Tridemethylsciadopitysin 3',8-Bi[4',5,7-trihydroxyflavone] 8-(5-(5,7-dihydroxy-4-oxo-4H-1-benzopyran-2-yl)-2-hydroxyphenyl)-5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-1-benzopyran-4-one 9I1VC79L77 AN-49542 CS-4945 HY-N0662 MolPort-001-741-078 SCHEMBL312563 YUSWMAULDXZHPY-UHFFFAOYSA-N 4H-1-Benzopyran-4-one, 8-(5-(5,7-dihydroxy-4-oxo-4H-1-benzopyran-2-yl)-2-hydroxyphenyl)-5,7-dihydroxy-2-(4-hydroxyphenyl)- 8-[5-(5,7-dihydroxy-4-oxo-4H-chromen-2-yl)-2-hydroxyphenyl]-5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one AKOS015896819 C-23136 Didemethyl-ginkgetin LMPK12040009 NSC 295677 SR-01000721725-2 [ Show all ]
Inchi Key	YUSWMAULDXZHPY-UHFFFAOYSA-N
Inchi ID	InChI=1S/C30H18O10/c31-15-4-1-13(2-5-15)24-12-23(38)29-21(36)10-20(35)27(30(29)40-24)17-7-14(3-6-18(17)33)25-11-22(37)28-19(34)8-16(32)9-26(28)39-25/h1-12,31-36H
PubChem CID	5281600
ChEMBL	CHEMBL63354
IUPHAR	N/A
BindingDB	N/A
DrugBank	N/A
Structure SDF download
Lipinski's druglikeness	This ligand has more than 5 hydrogen bond donor. This ligand is heavier than 500 daltons.

Known GPCRs

You can:

Click GLASS IDs to check the association information.
Click protein names to check details of the GPCRs.
Download a TSV version of all interaction information.

GLASS ID	Name	UniProt	Gene	Species	Length
419766	5-hydroxytryptamine receptor 1A	P08908	HTR1A	Homo sapiens (Human)	422
419790	5-hydroxytryptamine receptor 1B	P28222	HTR1B	Homo sapiens (Human)	390
419773	5-hydroxytryptamine receptor 1D	P28221	HTR1D	Homo sapiens (Human)	377
419776	5-hydroxytryptamine receptor 1D	P79400	HTR1D	Sus scrofa (Pig)	291
419788	5-hydroxytryptamine receptor 2C	P28335	HTR2C	Homo sapiens (Human)	458
419789	5-hydroxytryptamine receptor 5A	P47898	HTR5A	Homo sapiens (Human)	357
419770	5-hydroxytryptamine receptor 6	P50406	HTR6	Homo sapiens (Human)	440
419786	5-hydroxytryptamine receptor 7	P34969	HTR7	Homo sapiens (Human)	479
419777	Alpha-1A adrenergic receptor	P35348	ADRA1A	Homo sapiens (Human)	466
419784	Alpha-1B adrenergic receptor	P35368	ADRA1B	Homo sapiens (Human)	520
419785	Alpha-2A adrenergic receptor	P08913	ADRA2A	Homo sapiens (Human)	450
419792	Alpha-2B adrenergic receptor	P18089	ADRA2B	Homo sapiens (Human)	450
419779	Alpha-2C adrenergic receptor	P18825	ADRA2C	Homo sapiens (Human)	462
419781	D(1A) dopamine receptor	P21728	DRD1	Homo sapiens (Human)	446
419771	D(1B) dopamine receptor	P21918	DRD5	Homo sapiens (Human)	477
419791	D(3) dopamine receptor	P35462	DRD3	Homo sapiens (Human)	400
419775	Delta-type opioid receptor	P79291	OPRD1	Sus scrofa (Pig)	228
419778	Delta-type opioid receptor	P41143	OPRD1	Homo sapiens (Human)	372
419780	Glucagon-like peptide 1 receptor	P43220	GLP1R	Homo sapiens (Human)	463
419768	Kappa-type opioid receptor	P41145	OPRK1	Homo sapiens (Human)	380