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GPCR-RD is a database for experimental restaints of GPCRs. Although no solved X-ray or NMR structure is available for most GPCR sequences, numerous experiments have been performed on GPCRs to identify the critical residues and motifs. Experimental restraints were systematically collected from the literature using an automated text mining algorithm combined with manual validation, with the purpose of assisting GPCR 3-D structure modeling and function annotation. The GPCR-RD data are useful for GPCR 3D structure modeling, such as the GPCR-I-TASSER algorithm. The flow chart below summarizes the procedure for the extraction of experimental data and spatial restraints from literature and other resources.

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11002 entries in GPCR-RD.
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GPCR-RD: GPCR experimental restaint database
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Swiss-Prot ID Experimental Data Swiss-Prot ID Experimental Data Swiss-Prot ID Experimental Data
gabr1_rat C245A gabr1_rat C245S gabr1_rat S246A
gabr1_rat S246C gabr1_rat S246N gabr1_rat S246P
gabr1_rat S246T gabr1_rat S247A gabr1_rat S247C
gabr1_rat S249A gabr1_rat T250A gabr1_rat S265A
gabr1_rat Y266F gabr1_rat S268A gabr1_rat S269A
gabr1_rat S270A gabr1_rat T310A gabr1_rat Q312A
gabr1_rat Q313A gabr1_rat T314A gabr1_rat T315A
gabr1_rat T315C gabr1_rat E316A gabr1_rat E316C
gabr1_rat F365A gabr1_rat Y366A gabr1_rat E367A
gabr1_rat E458A gabr1_rat E459A gabr1_rat T460A
gabr1_rat F463A gabr1_rat Q464A gabr1_rat E465A
gabr1_rat Y470A gabr1_rat Y470F gabr1_rat D471A
gabr1_rat D471E boss_drovi K39A ste2_yeast S7K
ste2_yeast L8P ste2_yeast Q21R ste2_yeast N25Q
ste2_yeast N32Q ste2_yeast M54E ste2_yeast M54I
ste2_yeast M54T ste2_yeast M54V ste2_yeast F55L
ste2_yeast F55V ste2_yeast G56A ste2_yeast R58G
ste2_yeast R58H ste2_yeast C59I ste2_yeast G60A
ste2_yeast A62L ste2_yeast T65P ste2_yeast W70P
ste2_yeast S73P ste2_yeast N84S ste2_yeast H94L
ste2_yeast H94R ste2_yeast H94Y ste2_yeast S95H
ste2_yeast Y98H ste2_yeast F119L ste2_yeast F119S
ste2_yeast A140P ste2_yeast S141P ste2_yeast I142N
ste2_yeast E143K ste2_yeast T144A ste2_yeast T144P
ste2_yeast S145L ste2_yeast S145T ste2_yeast L146P
ste2_yeast L146Q ste2_yeast L146R ste2_yeast V147A
ste2_yeast Q149I ste2_yeast Q149N ste2_yeast Q149P
ste2_yeast Q149R ste2_yeast I150R ste2_yeast I153F
ste2_yeast I153N ste2_yeast F154L ste2_yeast I175V
ste2_yeast Y181N ste2_yeast T199C ste2_yeast Q200C
ste2_yeast D201C ste2_yeast K202C ste2_yeast Y203C


Reference:

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