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BioLiP E. coli GLASS GPCR-HGmod GPCR-RD GPCR-EXP TM-fold DECOYS POTENTIAL RW/RWplus HPSF THE-DB CASP7 CASP8 CASP9 CASP10 CASP11 CASP12 CASP13

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GPCR

NameGlucagon receptor
SpeciesRattus norvegicus (Rat)
GeneGcgr
SynonymGGR
GL-R
glucagon receptor
GR
DiseaseN/A for non-human GPCRs
Length485
Amino acid sequenceMLLTQLHCPYLLLLLVVLSCLPKAPSAQVMDFLFEKWKLYSDQCHHNLSLLPPPTELVCNRTFDKYSCWPDTPPNTTANISCPWYLPWYHKVQHRLVFKRCGPDGQWVRGPRGQSWRDASQCQMDDDEIEVQKGVAKMYSSYQVMYTVGYSLSLGALLLALVILLGLRKLHCTRNYIHGNLFASFVLKAGSVLVIDWLLKTRYSQKIGDDLSVSVWLSDGAVAGCRVATVIMQYGIIANYCWLLVEGVYLYSLLSITTFSEKSFFSLYLCIGWGSPLLFVIPWVVVKCLFENVQCWTSNDNMGFWWILRIPVLLAILINFFIFVRIIHLLVAKLRAHQMHYADYKFRLARSTLTLIPLLGVHEVVFAFVTDEHAQGTLRSTKLFFDLFFSSFQGLLVAVLYCFLNKEVQAELLRRWRRWQEGKALQEERMASSHGSHMAPAGTCHGDPCEKLQLMSAGSSSGTGCEPSAKTSLASSLPRLADSPT
UniProtP30082
Protein Data BankN/A
GPCR-HGmod modelN/A
3D structure modelNo available structures or models
BioLiPN/A
Therapeutic Target DatabaseN/A
ChEMBLCHEMBL4720
IUPHAR251
DrugBankN/A

Known ligands

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Total entries: 127
Page:  / 2 

GLASS IDMoleculeFormulaMolecular weightH-bond acceptor / donorXlogPLipinski's druglikeness
11832D structurec[Asp9, Lys12,] glucagon-NH2C153H224N44O47S3463.852 / 54-13.7No
51022D structureCHEMBL265503C55H71N11O19S21254.3521 / 17-1.0No
60972D structureCHEMBL265501C54H75N11O15S21182.3818 / 17-2.4No
90832D structureCHEMBL415177C123H182N36O422837.0247 / 45-18.0No
113902D structureCID 77078079C156H230N44O47S3505.8853 / 52-15.4No
4424522D structureCHEMBL3359004C16H12N2O4296.2824 / 22.5Yes
4429422D structureCHEMBL3326178C18H13N3O6367.3176 / 33.4Yes
333602D structureCID 44319559C143H214N42O47S3305.5953 / 52-19.5No
369032D structureGRA EX-25C29H36F3N3O5563.6188 / 35.8No
404852D structureBDBM50059363C142H217N41O47S3282.652 / 53-18.3No
4434992D structureCHEMBL3326184C18H12ClN3O6401.7596 / 34.0Yes
4435582D structureCHEMBL3326183C18H12FN3O6385.3077 / 33.5Yes
495092D structureCID 44319561C138H210N40O46S3197.4951 / 50-19.2No
501482D structure643011-22-7C27H21ClF3N3O3S559.9889 / 26.4No
518132D structureBDBM50098567C125H184N32O33S2695.137 / 39-5.0No
566482D structureBDBM50098574C127H182N32O32S2701.136 / 38-4.5No
594592D structureCID 44292844C154H224N40O46S3403.7850 / 49-11.2No
602162D structureCID 44335736C157H230N44O48S3533.8954 / 52-15.8No
646492D structureMK 0893C32H27Cl2N3O4588.4855 / 26.8No
4443002D structureGlucagon(10-20)amideC60H96N20O181385.5522 / 23-9.2No
4446982D structureCHEMBL3326187C22H21N3O6423.4256 / 35.3No
4448042D structureCHEMBL3326164C24H18N2O3382.4193 / 25.0Yes
798172D structureCHEMBL557974C22H24Cl2N4415.3624 / 05.6No
800502D structureCHEMBL2372773C153H224N42O47S3435.7852 / 51-16.4No
800512D structureCHEMBL266412C153H224N42O47S3435.7852 / 51-16.4No
830442D structureCID 44293064C154H226N40O47S3421.7952 / 50-15.6No
5600282D structureCHEMBL107070C18H13ClN2O3340.7634 / 34.0Yes
910672D structureCHEMBL442499C150H222N42O47S3397.7352 / 52-17.4No
945702D structureBDBM50104042C149H214N42O48S33457.7855 / 53-13.0No
4457442D structureCHEMBL3326165C24H18N2O4398.4184 / 34.7Yes
1071112D structureBDBM50104032C152H221N43O47S33498.8755 / 53-15.0No
1085412D structureCID 44278164C115H172N32O33S2562.8937 / 37-9.1No
1095142D structureCID 44292665C153H224N44O47S3463.852 / 52-14.5No
1096862D structureCID 44278221C123H180N32O33S2667.0437 / 37-6.9No
1150182D structureaminothiazole, 10C30H27Cl2N3O3S580.5246 / 27.5No
4462362D structureCHEMBL3325456C21H19N3O6409.3986 / 34.8Yes
1196462D structureCHEMBL152640C28H26N4O2450.5424 / 25.9No
1248262D structureCID 44335779C149H216N42O48S33459.7955 / 53-14.7No
4466202D structureCHEMBL3326175C24H17N3O6443.4156 / 35.0Yes
1279752D structureCID 44319558C138H209N39O47S3198.4852 / 50-18.5No
1287182D structureCHEMBL412352C145H219N43O47S3348.6653 / 52-19.3No
1290112D structureglucagon receptor antagonists-4C26H28F3N3O4503.5228 / 25.0No
1324212D structureCHEMBL1644183C27H20Cl2F3N3O4578.3698 / 26.4No
1391562D structureCHEMBL268583C165H226N36O553593.8260 / 52-15.9No
4472262D structureCHEMBL3326172C24H17ClN2O4432.864 / 35.3No
4478132D structureCHEMBL3326170C23H17N3O4399.4064 / 33.0Yes
4483222D structureCHEMBL3326179C19H15N3O6381.3446 / 33.8Yes
1744262D structureaminothiazole, 16C27H21ClF3N3O3S559.9889 / 26.4No
1752182D structureCID 44335967C152H223N43O47S33500.8955 / 53-16.2No
4487062D structureCHEMBL28541C35H50N8O10S2806.95113 / 13-1.4No
1797652D structureCID 77077841C153H224N44O47S3463.852 / 52-15.1No
4489402D structureCHEMBL3326166C24H18N2O4398.4184 / 34.7Yes
4492332D structureCHEMBL3326180C19H15N3O6381.3446 / 33.8Yes
4495402D structureCHEMBL3326186C21H19N3O6409.3986 / 34.5Yes
2009822D structureCHEMBL429362C153H225N43O49S3482.7955 / 53-17.7No
2009832D structureCID 102331734C153H225N43O49S3482.7987 / 590.8No
2013242D structureCID 71456274C153H223N41O46S3404.7751 / 50-15.3No
2013252D structureCID 71450989C153H223N41O46S3404.7751 / 50-15.3No
4497382D structureSCHEMBL3982429C24H18N2O5414.4175 / 44.3Yes
4505852D structureCHEMBL282363C35H48N8O10S2804.93513 / 11-0.9No
2270762D structureCID 44278463C121H176N32O33S2638.9937 / 37-7.5No
2303252D structureCHEMBL411904C86H127N25O301991.1134 / 33-15.0No
2394282D structureCHEMBL442492C165H224N36O493495.8155 / 50-11.0No
2575012D structureCHEMBL216417C51H68N10O16S21141.2818 / 17-0.9No
2590582D structureCID 77078086C150H219N43O49S33504.8357 / 55-19.2No
4521102D structureCHEMBL3326171C24H17FN2O4416.4085 / 34.8Yes
2654612D structureCID 44336110C154H225N41O48S3450.7953 / 51-15.4No
2676102D structureCID 71458083C147H219N41O46S3328.6751 / 50-16.9No
2676112D structureBDBM50407841C147H219N41O46S3328.6751 / 52-16.1No
4525162D structureSCHEMBL3976454C22H16N2O4372.384 / 24.1Yes
4525412D structureGlucagon(15-26)amideC67H102N22O191519.6936 / 280.4No
4528802D structureCHEMBL3326177C30H22N2O4474.5164 / 36.3No
2926562D structure[des-Phe6, Glu9] glucagonC139H211N39O47S3212.552 / 52-17.4No
3065052D structureCHEMBL2369990C148H221N41O47S3358.752 / 51-17.5No
3065062D structureCID 44278168C148H221N41O47S3358.752 / 51-17.5No
3072462D structureCHEMBL267646C55H73N11O19S21256.3721 / 19-2.0No
4541842D structureCHEMBL3326181C19H15N3O6381.3446 / 33.8Yes
3145192D structureCHEMBL408316C54H73N11O15S21180.3618 / 15-1.9No
4541942D structureGlucagon(5-16)amideC64H92N14O231425.5225 / 23-9.7No
3183862D structureAc-glucagon(6-29)amideC135H198N36O41S3013.3473 / 505.3No
3183942D structureCHEMBL413666C153H223N41O47S3420.7752 / 51-15.7No
3183952D structureCHEMBL2369127C153H223N41O47S3420.7752 / 51-15.7No
4545152D structureCHEMBL3326185C20H17N3O6395.3716 / 34.2Yes
3238912D structureCID 44278464C123H176N32O31S2631.0135 / 35-5.9No
3242592D structureaminothiazole, 6C34H26F3N3O4S629.65410 / 27.7No
3313862D structureCHEMBL152765C27H27N3O5473.5297 / 25.3No
3370062D structureCHEMBL266166C55H76N12O18S21257.421 / 20-5.6No
3430812D structureCHEMBL3037804C154H225N41O46S3418.7951 / 50-15.0No
3433832D structureCHEMBL557974C22H25Cl3N4451.824 / 1N/AN/A
4553872D structureAc-glucagon(6-14)amideC55H77N11O171164.2818 / 17-3.9No
3447422D structureCID 77078081C153H227N43O47S33516.9355 / 54-16.6No
3475482D structureCHEMBL412578C51H66N10O16S21139.2618 / 150.1No
3477122D structureBDBM50104035C151H228N44O47S3443.8153 / 54-16.5No
3508392D structureCID 44335807C150H217N43O49S33502.8257 / 53-18.7No
3524972D structureaminothiazole, 19C28H21F6N3O4S609.54313 / 27.0No
3527172D structureglucagon 1-6C29H41N9O10675.712 / 11-6.1No
4558002D structureGlucagon(1-11)amideC52H73N15O201228.2422 / 21-10.4No
3555802D structureCHEMBL386446C30H29Cl2N3O4566.4794 / 35.9No
3619842D structureBDBM50059358C148H221N41O48S3374.753 / 54-17.1No
3661622D structureCID 44336094C153H225N43O47S33514.9255 / 52-15.0No

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